Certificate of Analysis

 

Product Name: WAY-100635 Maleate
Catalog Number: M3481
CAS Number: 1092679-51-0

Physical and Chemical Properties
Formula: C25H34N4O2.C4H4O4
Molecular Weight: 538.64
Solubility: DMSO ≥ 100 mg/mL; Water 20 mg/mL
Storage: -20°C, dry, sealed
Chemical Structure: WAY-100635 Maleate Structure
Analytical Data
QC Standard: >99.0%
H-NMR: Consistent with structure
Product Information
Description: WAY-100635 maleate is a potent, selective 5-HT1A receptor antagonist with an IC50 value of 0.91 nM, a Ki value of 0.39 nM, and a pIC50 of 8.87, which is more than 100-fold more selective than for use at the other 5-HT receptor subtypes and major neurotransmitter receptors. In addition, WAY-100635 maleate is a potent dopamine D4 receptor agonist.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.