Certificate of Analysis

 

Product Name: TGR5 Receptor Agonist
Catalog Number: M2588
CAS Number: 1197300-24-5

Physical and Chemical Properties
Formula: C18H14Cl2N2O2
Molecular Weight: 361.22
Solubility: DMSO ≥ 30 mg/mL
Storage: Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Chemical Structure: TGR5 Receptor Agonist Structure
Analytical Data
QC Standard: >99%
H-NMR: Consistent with structure
Product Information
Description: TGR5 Receptor Agonist is a potent TGR5(GPCR19) agonist which showed improved potency in the U2-OS cell assay (pEC50 = 6.8) and in melanophore cells (pEC50 = 7.5).
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.