Certificate of Analysis

 

Catalog Number: M2735
Product Name: GSK2656157
CAS Number: 1337532-29-2

Physical and Chemical Properties
Formula: C23H21FN6O
Molecular Weight: 416.45
Solubility: DMSO 20 mg/mL
Long-term Storage: at -20℃
Chemical Structure: GSK2656157 Structure
Analytical Data
HPLC: Shows Min >99% purity
H-NMR: Consistent with structure
Product Information
Description: GSK2656157 is an ATP-competitive and highly selective inhibitor of PERK with IC50 of 0.9 nM, 500-fold greater against a panel of 300 kinases.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials at -20°C or below and used within 1 month.