Certificate of Analysis

 

Catalog Number: M2096
Product Name: GSK1210151A
CAS Number: 1300031-49-5

Physical and Chemical Properties
Formula: C23H21N5O3
Molecular Weight: 415.44
Solubility: DMSO 80 mg/mL
Long-term Storage: at -20℃
Chemical Structure: GSK1210151A Structure
Analytical Data
HPLC: Shows Min >99% purity
H-NMR: Consistent with structure
Product Information
Description: GSK1210151A (I-BET151) is an inhibitor of the BET family with IC50 of 0.5 μM, 0.25 μM and 0.79 μM for BRD2, BRD3 and BRD4, respectively.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials at -20°C or below and used within 1 month.