Certificate of Analysis

 

Product Name: Batefenterol (GSK961081)
Catalog Number: M5239
CAS Number: 743461-65-6

Physical and Chemical Properties
Formula: C40H42ClN5O7
Molecular Weight: 740.25
Solubility: DMSO 90 mg/mL
Storage: Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Chemical Structure: Batefenterol (GSK961081) Structure
Analytical Data
QC Standard: >98%
H-NMR: Consistent with structure
Product Information
Description: Batefenterol (GSK961081;TD-5959) is a novel muscarinic receptor antagonist and β2-adrenoceptor agonist; displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor with Ki values of 1.4, 1.3 and 3.7 nM, respectively.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.