Certificate of Analysis

 

Product Name: GLPG1690
Catalog Number: M6287
CAS Number: 1628260-79-6

Physical and Chemical Properties
Formula: C30H33FN8O2S
Molecular Weight: 588.7
Solubility: 10 mM in DMSO
Storage: Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Chemical Structure: GLPG1690 Structure
Analytical Data
QC Standard: 98.35%
H-NMR: Consistent with structure
Product Information
Description: GLPG1690 (Ziritaxestat) is a first-in-class autotaxin (ATX) inhibitor, with IC50 of 131 nM and Ki of 15 nM.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details.