Certificate of Analysis

 

Catalog Number: M6158
Product Name: ARQ-087
CAS Number: 1234356-69-4

Physical and Chemical Properties
Formula: C29H29FN4O
Molecular Weight: 468.57
Solubility: 10 mM in DMSO
Long-term Storage: at -20℃
Chemical Structure: ARQ-087 Structure
Analytical Data
HPLC: Shows Min >99% purity
H-NMR: Consistent with structure
Product Information
Description: ARQ 087 is a novel, ATP competitive, small molecule, multi-kinase inhibitor with potent in vitro and in vivo activity against FGFR addicted cell lines and tumors. ARQ 087 exhibited IC50 values of 1.8 nM for FGFR2, and 4.5 nM for FGFR1 and 3.
   
Stability and Solubility Advice: Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide.
We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials at -20°C or below and used within 1 month.